Life Science

Life Science

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  • Mericitabine | HY-10240

    Mericitabine | HY-10240

    Gentaur

    Mericitabine | HY-10240 Mericitabine (RG 7128; R-7128) is a nucleoside inhibitor of the HCV NS5B polymerase that acts as an RNA chain terminator and prevents elongation of RNA transcripts during replication. IC50 & Target : HCV NS5B polymerase In...
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  • Danoprevir | HY-10238

    Danoprevir | HY-10238

    Gentaur

    Danoprevir | HY-10238 Danoprevir (ITMN-191) is an orally active NS3/4A protease inhibitor for hepatitis C virus (HCV) with an IC50 of 0.29 nM and is selective for NS3/4A over a panel of 53 proteases (IC50 higher than 10 μM). Danoprevir (ITMN-191)...
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  • Boceprevir | HY-10237

    Boceprevir | HY-10237

    Gentaur

    Boceprevir | HY-10237 Boceprevir (EBP 520) is a potent, highly selective, orally bioavailable HCV NS3 protease inhibitor with a Ki of 14 nM in both enzyme assay and an EC90 of 350 nM in cell-based replicon assay. Boceprevir inhibits SARS-CoV-2 3CLpro...
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  • Telaprevir | HY-10235

    Telaprevir | HY-10235

    Gentaur

    Telaprevir | HY-10235 Telaprevir (VX-950) is a highly selective, reversible, and potent peptidomimetic inhibitor of the HCV NS3-4A protease, the steady-state inhibitory constant (Ki) of Telaprevir is 7 nM against a genotype 1 (H strain) NS3 protease...
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  • Saracatinib | HY-10234

    Saracatinib | HY-10234

    Gentaur

    Saracatinib | HY-10234 Saracatinib (AZD0530) is a potent Src family inhibitor with IC50s of 2.7 to 11 nM for c-Src, Lck, c-YES, Lyn, Fyn, Fgr, and Blk. Saracatinib shows high selectivity over other tyrosine kinases[1]. IC50 & Target : IC50: 2.7 nM...
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  • PX-478 | HY-10231

    PX-478 | HY-10231

    Gentaur

    PX-478 | HY-10231 PX-478 is an orally active HIF-1α inhibitor with potent antitumor activities. PX-478 can cross the blood-brain barrier[1][2]. IC50 & Target : HIF-1α[1] In Vitro: PC3 and DU 145 cells express HIF-1α protein are...
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  • Midostaurin | HY-10230

    Midostaurin | HY-10230

    Gentaur

    Midostaurin | HY-10230 Midostaurin (PKC412; CGP 41251) is an orally active, reversible multi-targeted protein kinase inhibitor. Midostaurin inhibits PKCα/β/γ, Syk, Flk-1, Akt, PKA, c-Kit, c-Fgr, c-Src, FLT3, PDFRβ and VEGFR1/2 with...
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  • Mirdametinib | HY-10254

    Mirdametinib | HY-10254

    Gentaur

    Mirdametinib | HY-10254 Mirdametinib (PD0325901) is an orally active, selective and non-ATP-competitive MEK inhibitor with an IC50 of 0.33 nM. Mirdametinib exhibits a Kiapp of 1 nM against activated MEK1 and MEK2. Mirdametinib suppresses the expression...
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  • AG1024 | HY-10253

    AG1024 | HY-10253

    Gentaur

    AG1024 | HY-10253 AG1024 (Tyrphostin AG 1024) is a reversible, competitive and selective IGF-1R inhibitor with an IC50 of 7 μM. AG1024 inhibits phosphorylation of IR (IC50=57 μM). AG1024 induces apoptosis and has anti-cancer activity[1][2]. IC50...
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  • NVP-ADW742 | HY-10252

    NVP-ADW742 | HY-10252

    Gentaur

    NVP-ADW742 | HY-10252 NVP-ADW742 (ADW742) is an orally active, selective IGF-1R tyrosine kinase inhibitor with an IC50 of 0.17 μM. NVP-ADW742 inhibits insulin receptor (InsR) with an IC50 of 2.8 μM. NVP-ADW742 induces pleiotropic...
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  • AKT Kinase Inhibitor | HY-10249A

    AKT Kinase Inhibitor | HY-10249A

    Gentaur

    AKT Kinase Inhibitor | HY-10249A AKT Kinase Inhibitor is an Akt kinase inhibitor with anti-tumor activity[1]. IC50 & Target : Akt In Vitro: The effect of selective inhibition of Akt in proliferating cells expressing Trop-2 is studied. Akt inhibition,...
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  • GSK-690693 | HY-10249

    GSK-690693 | HY-10249

    Gentaur

    GSK-690693 | HY-10249 GSK-690693 is an ATP-competitive pan-Akt inhibitor with IC50s of 2 nM, 13 nM, 9 nM for Akt1, Akt2 and Akt3, respectively. GSK-690693 is also an AMPK inhibitor, affects Unc-51-like autophagy activating kinase 1 (ULK1) activity and...
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